Dissection of the dual function of the beta-subunit of protein kinase CK2 ('casein kinase-2'): a synthetic peptide reproducing the carboxyl-terminal domain mimicks the positive but not the negative effects of the whole protein

FEBS Lett. 1995 Apr 17;363(1-2):111-4. doi: 10.1016/0014-5793(95)00295-k.

Abstract

The dual function of the regulatory beta-subunit of protein kinase CK2 is highlighted by its ability to abolish calmodulin phosphorylation in contrast to its stimulatory effect on the phosphorylation of peptide substrates. Here we show that a synthetic peptide reproducing the C-terminal region of the beta-subunit (beta[170-215]) stimulates to a similar extent the phosphorylation of either the peptide substrate or calmodulin and also protects the catalytic alpha-subunit against thermal inactivation as efficiently as full-length beta-subunit. These data show that the positive and negative functions of the beta-subunit reside in physically separated domains and that the elements responsible for positive regulation are located in the C-terminal region.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Binding Sites
  • Calmodulin / metabolism
  • Casein Kinase II
  • Enzyme Stability
  • Hot Temperature
  • Liver / enzymology
  • Macromolecular Substances
  • Molecular Sequence Data
  • Peptide Fragments / chemistry
  • Peptide Fragments / metabolism*
  • Phosphorylation
  • Protein Serine-Threonine Kinases / chemistry
  • Protein Serine-Threonine Kinases / metabolism*
  • Rats
  • Regulatory Sequences, Nucleic Acid
  • Structure-Activity Relationship

Substances

  • Calmodulin
  • Macromolecular Substances
  • Peptide Fragments
  • Casein Kinase II
  • Protein Serine-Threonine Kinases