ErbB-3 mediates differential mitogenic effects of NDF/heregulin isoforms on mouse keratinocytes

Oncogene. 1995 Apr 6;10(7):1403-11.

Abstract

The family of Neu differentiation factors (NDFs, or heregulins) includes a dozen secreted glycoproteins, whose receptor binding domain displays two variants, alpha and beta, and they bind to two receptor tyrosine kinases, ErbB-3 and ErbB-4. Certain isoforms were reported to induce growth-arrest and differentiation of mammary tumor cells, while other breast cancer cell lines responded mitogenically. The present study addressed the biologic effects of various NDF isoforms on normal EGF-dependent epithelial cells, Balb/MK keratinocytes, that can undergo either proliferation or differentiation. We found that beta isoforms of NDF induced a mitogenic effect, that was significantly smaller than the maximal response to EGF. By contrast with NDF-beta, NDF-alpha isoforms exerted almost no mitogenic effect, but they were sufficient to maintain keratinocytes in culture. Consistent with their higher mitogenic potency, NDF-beta isoforms bound to Balb/MK cells with higher affinity (Kd = 2.2 nM) than alpha isoforms, however both groups shared their receptor, that we identified as ErbB-3. No transcript of ErbB-4 was detectable in the keratinocytes, but these cells express multiple NDF mRNAs and also ErbB-2. We conclude that different isoforms of NDF induce distinct growth regulatory effects on cultured keratinocytes, through direct interaction with ErbB-3.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Base Sequence
  • Cells, Cultured
  • DNA Primers / chemistry
  • ErbB Receptors / metabolism
  • ErbB Receptors / physiology*
  • Gene Expression
  • Glycoproteins / chemistry
  • Glycoproteins / pharmacology*
  • Humans
  • In Vitro Techniques
  • Keratinocytes / cytology*
  • Mice
  • Mice, Inbred BALB C
  • Mitogens / pharmacology*
  • Molecular Sequence Data
  • Neuregulins
  • Proto-Oncogene Proteins / physiology*
  • RNA, Messenger / metabolism
  • Receptor, ErbB-3
  • Receptor, ErbB-4
  • Tumor Cells, Cultured

Substances

  • DNA Primers
  • Glycoproteins
  • Mitogens
  • Neuregulins
  • Proto-Oncogene Proteins
  • RNA, Messenger
  • ERBB4 protein, human
  • ErbB Receptors
  • Erbb4 protein, mouse
  • Receptor, ErbB-3
  • Receptor, ErbB-4