Stereoselective suppression of neutrophil function by ketamine?

Immunopharmacol Immunotoxicol. 1995 Feb;17(1):91-107. doi: 10.3109/08923979509052723.

Abstract

The effects of the commercially available ketamine preparation (Ketanest), the ketamine racemate and of the two enantiomers, the R(-)-racemate and the S(+)-racemate, as well as its drug-free solvent were examined by N-formyl-methionyl-leucyl-phenylalanine-(FMLP)- and zymosan-induced oxygen radical production of polymorphonuclear cells (PMN). The racemate and the two enantiomers of ketamine suppressed FMLP- and zymosan-induced chemiluminescence of PMN in a dose-dependent fashion to the same extent. Therefore suppression of chemiluminescence of PMN by ketamine does not result from a specific receptor interaction.

MeSH terms

  • Cell-Free System
  • Humans
  • In Vitro Techniques
  • Ketamine / chemistry
  • Ketamine / pharmacology*
  • Luminescent Measurements
  • N-Formylmethionine Leucyl-Phenylalanine / pharmacology
  • Neutrophils / drug effects*
  • Neutrophils / metabolism
  • Reactive Oxygen Species / metabolism
  • Stereoisomerism
  • Zymosan / pharmacology

Substances

  • Reactive Oxygen Species
  • N-Formylmethionine Leucyl-Phenylalanine
  • Ketamine
  • Zymosan