Engineering aspartic proteases to probe structure and function relationships

Curr Opin Biotechnol. 1994 Aug;5(4):422-7. doi: 10.1016/0958-1669(94)90052-3.

Abstract

Recently, protein engineering has been used to interconvert homodimeric and homologous single-chain aspartic proteases, with some success. The independent folding of the domains of these proteases has also permitted the engineering of domain-rearranged protease zymogens and the use of individual domains as probes for structural denaturation. In addition, site-directed mutagenesis has provided insights into the catalytic mechanism and specificity of this family of proteases.

Publication types

  • Review

MeSH terms

  • Aspartic Acid Endopeptidases / genetics*
  • Aspartic Acid Endopeptidases / metabolism*
  • Biological Evolution
  • Models, Molecular
  • Protein Engineering
  • Structure-Activity Relationship
  • Substrate Specificity

Substances

  • Aspartic Acid Endopeptidases