p53 transcriptional activation mediated by coactivators TAFII40 and TAFII60

Science. 1995 Jan 6;267(5194):100-4. doi: 10.1126/science.7809597.

Abstract

The tumor suppressor protein p53 is a transcriptional regulator that enhances the expression of proteins that control cellular proliferation. The multisubunit transcription factor IID (TFIID) is thought to be a primary target for site-specific activators of transcription. Here, a direct interaction between the activation domain of p53 and two subunits of the TFIID complex, TAFII40 and TAFII60, is reported. A double point mutation in the activation domain of p53 impaired the ability of this domain to activate transcription and, simultaneously, its ability to interact with both TAFII40 and TAFII60. Furthermore, a partial TFIID complex containing Drosophila TATA binding protein (dTBP), human TAFII250, dTAFII60, and dTAFII40 supported activation by a Gal4-p53 fusion protein in vitro, whereas TBP or a subcomplex lacking TAFII40 and TAFII60 did not. Together, these results suggest that TAFII40 and TAFII60 are important targets for transmitting activation signals between p53 and the initiation complex.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Sequence
  • DNA-Binding Proteins / metabolism
  • Drosophila Proteins*
  • HeLa Cells
  • Histone Acetyltransferases
  • Humans
  • Molecular Sequence Data
  • Nuclear Proteins / metabolism
  • Point Mutation
  • Recombinant Fusion Proteins / metabolism
  • TATA-Binding Protein Associated Factors*
  • TATA-Box Binding Protein
  • Trans-Activators / metabolism*
  • Transcription Factor TFIID*
  • Transcription Factors / metabolism*
  • Transcriptional Activation*
  • Tumor Suppressor Protein p53 / genetics
  • Tumor Suppressor Protein p53 / metabolism*

Substances

  • DNA-Binding Proteins
  • Drosophila Proteins
  • Nuclear Proteins
  • Recombinant Fusion Proteins
  • TATA-Binding Protein Associated Factors
  • TATA-Box Binding Protein
  • Trans-Activators
  • Transcription Factor TFIID
  • Transcription Factors
  • Tumor Suppressor Protein p53
  • e(y)1 protein, Drosophila
  • Histone Acetyltransferases
  • TATA-binding protein associated factor 250 kDa