The minimal active domain of the mouse ras exchange factor CDC25Mm

Biochem Biophys Res Commun. 1995 Jan 5;206(1):253-9. doi: 10.1006/bbrc.1995.1035.

Abstract

The minimal active domain of the mouse CDC25Mm, a GDP/GTP exchange factor (GEF) active on H-ras protein, was determined by constructing several deletion mutants of the C-terminal domain of the protein. The functional activity of these fragments was analyzed for the ability to complement the yeast temperature sensitive mutation cdc25-1 and to catalyze the GDP/GTP exchange on Ras proteins in vitro. A C-terminal domain of 256 residues (CDC25Mm 1005-1260) was sufficient for full biological activity in vivo. Deletion of 27 C-terminal amino acids (CDC25Mm 1005-1233) abolished the complementing activity while deletion of 25 N-terminal residues (CDC25Mm 1030-1260 corresponding to the most conserved domain) led to a complete loss of expression. The results in vivo were supported by experiments in vitro. Highly purified CDC25Mm 1005-1260, expressed in E. coli using the pMAL system, enhanced the GDP release from both H-ras p21 and S. cerevisiae Ras2p and its activity was nearly as high as that of CDC25Mm 974-1260. Comparison with the Cdc25p protein yielded further evidence that the minimal active domain of CDC25Mm is shorter than the yeast one.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Cycle Proteins*
  • Fungal Proteins / biosynthesis
  • Fungal Proteins / chemistry*
  • Fungal Proteins / metabolism*
  • Gene Deletion
  • Genetic Complementation Test
  • Guanine Nucleotide Exchange Factors
  • Guanosine Diphosphate / metabolism
  • Kinetics
  • Mice
  • Mutagenesis
  • Plasmids
  • Polymerase Chain Reaction
  • Proteins / chemistry*
  • Proto-Oncogene Proteins p21(ras) / metabolism
  • Restriction Mapping
  • Saccharomyces cerevisiae / genetics
  • Saccharomyces cerevisiae / metabolism*
  • Saccharomyces cerevisiae Proteins
  • Structure-Activity Relationship
  • ras Guanine Nucleotide Exchange Factors
  • ras-GRF1*

Substances

  • CDC25 protein, S cerevisiae
  • Cell Cycle Proteins
  • Fungal Proteins
  • Guanine Nucleotide Exchange Factors
  • Proteins
  • Saccharomyces cerevisiae Proteins
  • ras Guanine Nucleotide Exchange Factors
  • ras-GRF1
  • Guanosine Diphosphate
  • Proto-Oncogene Proteins p21(ras)