Calcium ion binding to thrombospondin 1

J Biol Chem. 1995 Jan 27;270(4):1729-33. doi: 10.1074/jbc.270.4.1729.

Abstract

We have quantified the binding of Ca2+ to platelet thrombospondin 1 (TSP1) using equilibrium dialysis with 45CaCl2. Ca2+ binding to TSP1 was found to be cooperative with 10% occupancy at 15-20 microM CaCl2, 90% occupancy at 100 microM CaCl2, and a Hill coefficient of 2.4 +/- 0.2 The average apparent Kd was 52 +/- 5 microM. Maximum binding, assuming Mr = 450,000 and epsilon = 0.918 (A280/mg/ml), was 35 +/- 3 Ca2+/TSP1. This value is close to the 33 sites (11 per subunit) predicted based on homology of the epidermal growth factor (1 site) and aspartate-rich (10 sites) regions to known Ca2+ binding sequences. Ca2+ protected the aspartate-rich region from trypsin proteolysis, but not until nearly all of the Ca2+ binding sites were filled. At lower occupancy of Ca2+ binding sites, several limited tryptic digest products were obtained. This finding and the previous demonstration of extensive thiol-disulfide isomerization within the aspartate-rich regions suggest that subregions of the aspartate-rich region are stabilized in different conformers. Zn2+, Cu2+, Mn2+, Mg2+, Co2+, Cd2+, and Ba2+ were tested for their ability to modulate Ca2+ binding and protease sensitivity of TSP1. Zn2+ inhibited 40% of the Ca2+ binding but neither protected TSP1 from trypsin proteolysis, nor labilized TSP1 toward trypsin proteolysis. These results provide direct evidence for high capacity, cooperative and specific binding of Ca2+ to conformationally labile aspartate-rich repeats of TSP1.

Publication types

  • Comparative Study
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Blood Platelets / metabolism*
  • Calcium / metabolism*
  • Calcium Radioisotopes
  • Cations, Divalent / pharmacology
  • Consensus Sequence
  • Humans
  • Kinetics
  • Membrane Glycoproteins / blood*
  • Membrane Glycoproteins / chemistry
  • Membrane Glycoproteins / isolation & purification
  • Molecular Sequence Data
  • Peptide Fragments / chemistry
  • Peptide Fragments / isolation & purification
  • Peptide Fragments / metabolism
  • Protein Binding
  • Repetitive Sequences, Nucleic Acid
  • Sequence Homology, Amino Acid
  • Thrombospondins
  • Trypsin / metabolism
  • Zinc / pharmacology

Substances

  • Calcium Radioisotopes
  • Cations, Divalent
  • Membrane Glycoproteins
  • Peptide Fragments
  • Thrombospondins
  • Trypsin
  • Zinc
  • Calcium