Ion-transporting activity in the murine colonic epithelium of normal animals and animals with cystic fibrosis

Pflugers Arch. 1994 Oct;428(5-6):508-15. doi: 10.1007/BF00374572.

Abstract

Electrogenic ion transport in the isolated colonic epithelium from normal and transgenic mice with cystic fibrosis (CF mice) has been investigated under short-circuit current (Isc) conditions. Normal tissues showed chloride secretion in response to carbachol or forskolin, which was sensitive to the Na-K-2Cl cotransport inhibitor, frusemide. Responses to both agents were maintained for at least 12 h in vitro, but the responses to carbachol changed in format throughout this period. By contrast CF colons failed to show the normal secretory responses to carbachol and forskolin, most preparations showing a decrease in Isc that was immediately reversed by frusemide. In CF colons addition of Ba2+ ions or tetraethylammonium (TEA+) to the apical bathing solution antagonised the reduction in Isc caused by the secretagogues. It is concluded that the reduction in Isc in CF colons is due to electrogenic K+ secretion and this was confirmed by flux studies using rubidium-86. In normal colons exposed to TEA+ the responses to forskolin were greater, but not significantly so, presumably because the minor K(+)-secretory responses are dominated by major chloride-secretory responses. Again rubidium-86 fluxes showed an increase of K+ secretion in normal colons receiving forskolin. Since the amiloride-sensitive current was not different in CF and normal colons there was no evidence that the CF mice were stressed in a way that increased mineralocorticoid levels and hence K+ secretion. Knowledge of the phenotype of the colonic epithelium of the CF mouse sets the baseline from which attempts at gene therapy for the gut must be judged.

MeSH terms

  • Amiloride / pharmacology
  • Animals
  • Biological Transport / drug effects
  • Carbachol / pharmacology
  • Colforsin / pharmacology
  • Colon / metabolism*
  • Cystic Fibrosis / metabolism*
  • Epithelium
  • Furosemide / pharmacology
  • Ions*
  • Mice
  • Mice, Inbred CFTR
  • Potassium / metabolism*
  • Rubidium Radioisotopes / metabolism
  • Tetraethylammonium
  • Tetraethylammonium Compounds / metabolism

Substances

  • Ions
  • Rubidium Radioisotopes
  • Tetraethylammonium Compounds
  • Colforsin
  • Tetraethylammonium
  • Amiloride
  • Furosemide
  • Carbachol
  • Potassium