Glucagon-like peptide-1 modulates Ca2+ current but not K+ATP current in intact mouse pancreatic B-cells

Biochem Biophys Res Commun. 1995 Feb 6;207(1):33-9. doi: 10.1006/bbrc.1995.1149.

Abstract

The influence of GLP-1 on electrical activity and ion currents of mouse pancreatic B-cells was studied with intracellular microelectrodes and the whole-cell configuration of the patch-clamp technique. In the presence of 15 mmol/l glucose 5, 50 and 100 nmol/l GLP-1 slightly increased electrical activity. This effect may be caused by the slowing of Ca2+ channel inactivation observed with GLP-1. Thus, changes in Ca2+ channel kinetics are suggested to contribute to the insulinotropic action of the hormone. The most prominent effect of GLP-1 on the membrane potential was the conversion of irregular electrical activity into regular oscillations of the membrane potential. At the threshold concentration for insulin secretion (7 mmol/l glucose) GLP-1 did not alter the membrane potential. Accordingly, in patch-clamp experiments GLP-1 had no effect on the whole-cell K+ATP current.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenosine Triphosphate / metabolism*
  • Animals
  • Calcium Channels / drug effects
  • Calcium Channels / physiology*
  • Female
  • Glucagon / pharmacology*
  • Glucagon-Like Peptide 1
  • Glucagon-Like Peptides
  • Glucose / pharmacology
  • In Vitro Techniques
  • Islets of Langerhans / drug effects
  • Islets of Langerhans / physiology*
  • Kinetics
  • Membrane Potentials / drug effects
  • Mice
  • Mice, Inbred Strains
  • Peptide Fragments / pharmacology*
  • Peptides / pharmacology
  • Potassium Channels / drug effects
  • Potassium Channels / physiology*
  • Protein Precursors / pharmacology*

Substances

  • Calcium Channels
  • Peptide Fragments
  • Peptides
  • Potassium Channels
  • Protein Precursors
  • glucagon-like peptide 1 (7-36)amide
  • Glucagon-Like Peptides
  • Glucagon-Like Peptide 1
  • Adenosine Triphosphate
  • Glucagon
  • Glucose
  • glucagon-like peptide 1 (7-37)