Effect of tetracyclines on collagenase activity in patients with recurrent aphthous ulcers

J Oral Pathol Med. 1994 Jul;23(6):269-72. doi: 10.1111/j.1600-0714.1994.tb00057.x.

Abstract

Human neutrophil-type (MMP-8) and fibroblast-type (MMP-1) interstitial collagenase, and their inhibition by tetracyclines in saliva from patients with recurrent aphthous ulcers (RAU) or aphthae, were studied by means of sodium dodecyl sulfate polyacrylamide gel electrophoresis (SDS-PAGE) and enzymological analyses. In the salivary specimens obtained from patients with aphthae, collagenase was found in endogenously active form and was predominantly of MMP-8 type. Topical rinsing treatment with chlortetracycline (Aureomycin) alleviated the discomfort caused by the lesions but did not reduce salivary collagenase amounts; however in vitro, doxycycline inhibited salivary collagenase totally.

Publication types

  • Clinical Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adolescent
  • Adult
  • Child
  • Chlortetracycline / administration & dosage
  • Chlortetracycline / therapeutic use*
  • Collagenases / metabolism
  • Doxycycline / pharmacology
  • Electrophoresis, Polyacrylamide Gel
  • Female
  • Fibroblasts / enzymology
  • Humans
  • Male
  • Matrix Metalloproteinase 1
  • Matrix Metalloproteinase 8
  • Matrix Metalloproteinase Inhibitors*
  • Middle Aged
  • Mouthwashes / therapeutic use
  • Neutrophils / enzymology
  • Recurrence
  • Saliva / enzymology
  • Stomatitis, Aphthous / drug therapy*
  • Stomatitis, Aphthous / enzymology*

Substances

  • Matrix Metalloproteinase Inhibitors
  • Mouthwashes
  • Collagenases
  • Matrix Metalloproteinase 8
  • Matrix Metalloproteinase 1
  • Doxycycline
  • Chlortetracycline