Constitutive expression of B-myb can bypass p53-induced Waf1/Cip1-mediated G1 arrest

Proc Natl Acad Sci U S A. 1994 Oct 11;91(21):10079-83. doi: 10.1073/pnas.91.21.10079.

Abstract

Overexpression of wild-type p53 protein has been shown to induce arrest in the G1 stage of the cell cycle and to transactivate expression of the gene that encodes the 21-kDa Waf1/Cip1 protein, a potent inhibitor of cyclin-dependent kinase activity. p53-dependent G1 arrest is accompanied by decreased expression of the B-myb gene, a relative of the c-myb cellular oncogene. In this study we show that B-myb expression is required for cells to progress from G1 into S phase and that high levels of ectopic B-myb expression uncoupled from cell cycle regulation rescues cells from p53-induced G1 arrest even in the presence of Waf1/Cip1 transactivation and inhibition of cyclin E/Cdk2 kinase activity. Cotransfection experiments with p53 expression plasmids and expression plasmids encoding in-frame deletion mutations in B-myb coding sequences indicate that the DNA-binding domain of the B-Myb protein is required for this activity. These results provide evidence of a bypass of p53-induced Waf1/Cip1-mediated cell cycle regulatory pathways by a member of the myb oncogene family.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Base Sequence
  • Blotting, Northern
  • Cell Cycle / drug effects
  • Cell Cycle / physiology*
  • Cell Cycle Proteins*
  • Cell Line
  • Cyclin-Dependent Kinase Inhibitor p21
  • Cyclins / metabolism*
  • DNA-Binding Proteins / biosynthesis
  • DNA-Binding Proteins / metabolism*
  • G1 Phase
  • Gene Expression*
  • Genes, p53
  • Humans
  • Molecular Sequence Data
  • Oligonucleotides, Antisense / pharmacology*
  • Oncogenes*
  • Osteosarcoma
  • Plasmids
  • Protein Kinase Inhibitors*
  • RNA, Messenger / analysis
  • RNA, Messenger / biosynthesis
  • Trans-Activators*
  • Transcription Factors / biosynthesis
  • Transcription Factors / metabolism*
  • Transfection
  • Tumor Cells, Cultured
  • Tumor Suppressor Protein p53 / metabolism*

Substances

  • CDKN1A protein, human
  • Cell Cycle Proteins
  • Cyclin-Dependent Kinase Inhibitor p21
  • Cyclins
  • DNA-Binding Proteins
  • MYBL2 protein, human
  • Oligonucleotides, Antisense
  • Protein Kinase Inhibitors
  • RNA, Messenger
  • Trans-Activators
  • Transcription Factors
  • Tumor Suppressor Protein p53