Role of protein kinase C in ras-mediated fos-expression

Adv Enzyme Regul. 1994:34:257-68. doi: 10.1016/0065-2571(94)90020-5.

Abstract

HC-11 mouse mammary epithelial cells stably transfected with a glucocorticoid-inducible Ha-ras construct encoding a transforming (val12) p21Ha-ras were cotransfected with a c-fos-CAT construct containing the human c-fos promoter up to position -711 and the CAT reporter gene. Expression of Ha-ras by dexamethasone leads to a transcriptional activation of the fos-CAT construct which was found to be sensitive to the PKC inhibitor ilmofosine (BM41440) and abrogated by PKC depletion following long-term exposure to TPA. The responsiveness to Ha-ras is retained if only the portion of the fos promoter covering the serum response element (SRE) and the adjacent fos AP-1 (FAP) site are put in front of a CAT gene linked to a thymidine kinase (TK) promoter. Further depletion of the FAP-site does not affect the inducibility by Ha-ras. Transcriptional activation of the SRE-FAP-TK-CAT as well as the SRE-TK-CAT constructs by Ha-ras is sensitive to the PKC-inhibitor ilmofosine (BM41440) and blocked by long-term exposure to TPA. Long-term exposure to TPA depletes cells of PKC alpha and significantly reduces the PKC epsilon levels. Long-term exposure in bryostatin 1 selectively depletes PKC alpha. Depletion of PKC alpha by bryostatin 1 does not reduce the transcriptional activation of the SRE-FAP-TK-CAT-construct by Ha-ras. It is concluded that (i) transforming Ha-ras induces c-fos in HC-11 cells via PKC (presumably epsilon), (ii) the signal is mediated to the serum response element (SRE) of the fos promoter and (iii) the fos AP-1 (FAP) site is not required for this mechanism.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Bryostatins
  • Cell Compartmentation
  • Cell Line
  • Epithelial Cells
  • Gene Expression Regulation* / drug effects
  • Isoenzymes / metabolism*
  • Lactones / pharmacology
  • Macrolides
  • Mammary Glands, Animal / cytology
  • Mice
  • Protein Kinase C / metabolism*
  • Proto-Oncogene Proteins c-fos / biosynthesis*
  • Recombinant Proteins / biosynthesis
  • Signal Transduction
  • Tetradecanoylphorbol Acetate / pharmacology
  • Transcription, Genetic
  • Transfection
  • ras Proteins / metabolism*

Substances

  • Bryostatins
  • Isoenzymes
  • Lactones
  • Macrolides
  • Proto-Oncogene Proteins c-fos
  • Recombinant Proteins
  • bryostatin 1
  • Protein Kinase C
  • ras Proteins
  • Tetradecanoylphorbol Acetate