Heterodimerization and deoxyribonucleic acid-binding properties of a retinoid X receptor-related factor

Endocrinology. 1994 Nov;135(5):2076-85. doi: 10.1210/endo.135.5.7956930.

Abstract

The extent thyroid hormone receptors (TRs) bind to AGGTCA-related motifs as monomers and/or homodimers, and as heterodimers with retinoid X receptors (RXRs) depends on the number, spacing, and orientation of these half-sites. Here we show that recombinant RXR alpha affects TR binding to DNA in diverse ways; it enhances recombinant TR beta 1 binding to four-nucleotide-spaced direct repeat and palindromes but not to inverted palindromes. We also used an endogenous factor termed RXR alpha-RF that cross-reacted with antibodies to RXR alpha and copurified and formed heterodimers on DNA with rat liver TRs (mostly TR beta 1 isoform), supporting the fact that endogenous TRs are commonly heterodimers. RXR alpha-RF formed, like recombinant RXR alpha, heterodimers on DNA with vitamin D and retinoic acid but not estrogen receptors. RXR alpha-RF differed from recombinant RXR alpha in that it provoked enhancement of TR beta 1 binding to DNA irrespective of half-site architecture, was resistant to heating to 50 C, and did not form heterodimers with recombinant TR alpha 2 on four-nucleotide-spaced direct repeat. The overall enhancement of TR-DNA recognition by endogenous RXR alpha-RF, not found in studies with recombinant RXR alpha, might exemplify properties acquired in vivo by endogenous RXRs; this could promote wider DNA recognition by TRs and expand the thyroid hormone transcriptional influence in the cell.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Base Sequence
  • DNA / analysis
  • DNA / genetics
  • DNA / metabolism*
  • Liver / chemistry
  • Liver / metabolism
  • Liver / ultrastructure
  • Molecular Sequence Data
  • Protein Binding
  • Protein Conformation
  • Rats
  • Receptors, Cytoplasmic and Nuclear / analysis*
  • Receptors, Cytoplasmic and Nuclear / metabolism
  • Receptors, Cytoplasmic and Nuclear / physiology*
  • Receptors, Retinoic Acid*
  • Receptors, Thyroid Hormone / analysis
  • Receptors, Thyroid Hormone / metabolism
  • Retinoid X Receptors
  • Transcription Factors / analysis*
  • Transcription Factors / metabolism
  • Transcription Factors / physiology*

Substances

  • Receptors, Cytoplasmic and Nuclear
  • Receptors, Retinoic Acid
  • Receptors, Thyroid Hormone
  • Retinoid X Receptors
  • Transcription Factors
  • DNA