An antitumor, branched (1-->3)-beta-D-glucan from a water extract of fruiting bodies of Cryptoporus volvatus

Carbohydr Res. 1994 Oct 3;263(1):111-21. doi: 10.1016/0008-6215(94)00156-1.

Abstract

A water-soluble, (1-->6)-branched (1-->3)-beta-D-glucan (H-3-B) was isolated from a hot-water extract of the fruiting bodies of the fungus, Cryptoporus volvatus (Basidiomycetes). Enzymatic analysis using exo-(1-->3)-beta-D-glucanase and methylation analysis indicated that this polysaccharide has a main chain composed of beta-(1-->3)-linked D-glucopyranosyl residues, and single, beta-(1-->6)-linked D-glucopyranosyl residues attached as side chains to, on average, every fourth sugar residue of the main chain. This structure was confirmed by 13C NMR spectra of the glucan in Me2SO-d6. The weight-average molecular weight (Mw) of H-3-B was determined to be 44.0 x 10(4) by gel permeation chromatography equipped with a low-angle laser-light-scattering photometer. The electron microscopic observations showed that H-3-B and its sonicated sample (S-H-3-B, Mw = 13.7 x 10(4)) can be described as linear worm-like chains. The mass per unit length for native and sonicated H-3-B was determined to be 1750 and 1780 g mol-1 nm-1, respectively, from the contour lengths obtained by electron microscopy and the molecular weights. These values are in good agreement with that expected for the triple stranded structure. A sample denatured in 0.1 M NaOH and subsequently renatured by neutralization showed a mixture of linear and cyclic structures, and larger aggregates with less well-defined morphology. The H-3-B and S-H-3-B had antitumor activity against the Sarcoma 180 tumor.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antineoplastic Agents / isolation & purification*
  • Antineoplastic Agents / pharmacology
  • Basidiomycota / chemistry*
  • Carbohydrate Conformation
  • Carbohydrate Sequence
  • Chromatography, Gel
  • Glucans / isolation & purification*
  • Glucans / pharmacology
  • Light
  • Magnetic Resonance Spectroscopy
  • Microscopy, Electron
  • Molecular Sequence Data
  • Molecular Weight
  • Plant Extracts / analysis*
  • Sarcoma 180 / drug therapy
  • Scattering, Radiation
  • Sizofiran / pharmacology
  • Water

Substances

  • Antineoplastic Agents
  • Glucans
  • Plant Extracts
  • Water
  • Sizofiran