Ligand binding characteristics of [3H] dihydroalprenolol in cerebral cortical membranes of young and old senescence-accelerated mouse

Comp Biochem Physiol C Comp Pharmacol Toxicol. 1993 Mar;104(3):423-6.

Abstract

1. The values of both Kd and Bmax of [3H] dihydroalprenolol binding in the cerebral cortical membranes of old-aged (12 month old) SAM-P/1 were not significantly different compared with those of young (2 month old) SAM-P/1. 2. The values of Ki of metoprolol in the young and old aged SAM were 119 +/- 39.5 nM and 157 +/- 55 nM, respectively. 3. The values of beta 1/beta 2 ratio of the young and old aged SAM were 1.67 +/- 0.15 and 1.64 +/- 0.13, respectively. 4. These results suggest that there were no significant changes of binding characteristics of beta 1 and beta 2 adrenoceptors during aging in the cerebral cortex of SAM.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aging / metabolism*
  • Animals
  • Cerebral Cortex / metabolism*
  • Dihydroalprenolol / metabolism*
  • Male
  • Metoprolol / pharmacology
  • Mice
  • Radioligand Assay
  • Receptors, Adrenergic, beta / metabolism*

Substances

  • Receptors, Adrenergic, beta
  • Dihydroalprenolol
  • Metoprolol