[The role of extracellular calcium in the vasoconstriction evoked by endothelin-1]

Biull Eksp Biol Med. 1993 Sep;116(9):258-60.
[Article in Russian]

Abstract

Some mechanisms responsible for extracellular Ca++ entry into rat aortic smooth muscle cells were studied in response to endothelin-1 (ET-1). Isometric tension of de-endothelialized aortic strips was recorded. It was shown that the calcium-free medium or nifedipine blockade of calcium entry diminished responses to ET-1 to 20-30% of the control levels. Depolarization of the specimens with hyperpotassium solution also reduced constriction almost by 50%. When sodium ions were replaced by NMDG in the medium, a response to ET-1 showed a 50% reduction. The findings suggest that the potential-dependent calcium channels of the L-type are involved in cellular calcium entry, the opening of the channels depending upon the entry of Na+.

Publication types

  • English Abstract

MeSH terms

  • Animals
  • Calcium / pharmacology*
  • Calcium / physiology
  • Calcium Channels / drug effects
  • Calcium Channels / physiology
  • Endothelins / pharmacology*
  • Endothelium, Vascular / physiology
  • In Vitro Techniques
  • Meglumine / pharmacology
  • Muscle Contraction / drug effects
  • Muscle Contraction / physiology
  • Muscle, Smooth, Vascular / drug effects
  • Muscle, Smooth, Vascular / physiology
  • Nifedipine / pharmacology
  • Phenylephrine / pharmacology
  • Rats
  • Rats, Wistar
  • Vasoconstriction / drug effects*
  • Vasoconstriction / physiology

Substances

  • Calcium Channels
  • Endothelins
  • Phenylephrine
  • Meglumine
  • Nifedipine
  • Calcium