Regulation of rat-kidney cortex fructose-1,6-bisphosphatase activity. I. Effects of fructose-2,6-bisphosphate and divalent cations

Int J Biochem. 1993 Dec;25(12):1963-8. doi: 10.1016/0020-711x(88)90332-1.

Abstract

1. The native rat-kidney cortex Fructose-1,6-BPase is differentially regulated by Mg2+ and Mn2+. 2. Mg2+ binding to the enzyme is hyperbolic and large concentrations of the cation are non-inhibitory. 3. Mn2+ produces a 10-fold rise in Vmax higher than Mg2+. [Mn2+]0.5 is much larger than [Mg2+]0.5. At elevated [Mn2+] inhibition is observed. 4. Mg2+ and Mn2+ produce antagonistic effects on the inhibition of the enzyme by high substrate. 5. Fru-2,6-P2 inhibits the enzyme by rising the S0.5 and favouring a sigmoidal kinetics. 6. The inhibition by Fru-2,6-P2 is released by Mg2+ and more powerfully by Mn2+ increasing the I0.5.

MeSH terms

  • Animals
  • Fructose-Bisphosphatase / antagonists & inhibitors
  • Fructose-Bisphosphatase / drug effects*
  • Fructosediphosphates / pharmacology*
  • Kidney Cortex / drug effects*
  • Kidney Cortex / enzymology
  • Kinetics
  • Magnesium / pharmacology*
  • Male
  • Manganese / pharmacology*
  • Rats
  • Rats, Wistar

Substances

  • Fructosediphosphates
  • Manganese
  • fructose 2,6-diphosphate
  • Fructose-Bisphosphatase
  • Magnesium