Molecular heterogeneity of the type I GABAA/benzodiazepine receptor complex

Eur J Pharmacol. 1994 Mar 15;267(1):123-8. doi: 10.1016/0922-4106(94)90233-x.

Abstract

We have investigated the presence of alpha 1, gamma 2 and beta 2-3 subunits as part of the type I (high affinity for [3H]zolpidem) GABAA/benzodiazepine receptor from rat cerebral cortex. Three subunit specific antibodies have been used (anti-alpha 1, to the C-terminal of rat alpha 1 subunit; anti-gamma 2, to the large intracellular loop of the gamma 2 subunit short form and the monoclonal 62-3G1, specific to beta 2-3 subunits) in immunoprecipitation experiments of the [3H]zolpidem binding activity or the 51,000 Da [3H]Ro 15-4513 photoaffinity labeled peptide (P51). The results indicated that alpha 1 subunit was present in the whole population (90%) of the GABAA/benzodiazepine receptors with high affinity for [3H]zolpidem. We cannot exclude the presence of other alpha subunits co-localized with alpha 1. On the one hand, 70-75% of type I GABAA/benzodiazepine receptor from rat cortex have co-existing alpha 1, beta 2-3 and gamma 2 subunits. We call this type Ia. On the other hand, 20-25% of the type I GABAA/benzodiazepine receptor complex should be constructed by the association of alpha 1 with subunits other than beta 2-3 and gamma 2. We call this type Ib. The identity of these subunits is currently unknown.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Benzodiazepines / metabolism*
  • Binding Sites
  • Cerebral Cortex / metabolism*
  • Precipitin Tests
  • Pyridines / metabolism*
  • Rats
  • Rats, Wistar
  • Receptors, GABA-A / chemistry*
  • Receptors, GABA-A / physiology
  • Zolpidem

Substances

  • Pyridines
  • Receptors, GABA-A
  • Benzodiazepines
  • Zolpidem