Effect of gangliosides on diacylglycerol content and molecular species in nerve from diabetic rats

Eur J Pharmacol. 1993 Aug 3;239(1-3):55-61. doi: 10.1016/0014-2999(93)90975-n.

Abstract

The effects of ganglioside treatment on 1,2-diacylglycerol content and on molecular species in 1,2-diacylglycerol, phosphatidic acid and total diacylglycerolipids, as well as Na+,K(+)-ATPase activity, were examined in sciatic nerves from streptozotocin-induced diabetic rats. Beginning 2 weeks after induction of diabetes, animals were administered mixed bovine brain gangliosides, AGF1, an inner ester derivative of this mixture, or saline for 5 weeks. The levels of 1,2-diacylglycerol and arachidonoyl-containing molecular species in age-matched non-diabetic animals were not affected by ganglioside treatment. In nerves from saline-treated diabetic animals, 1,2-diacylglycerol levels were not reduced, but both Na+,K(+)-ATPase activity and all arachidonyl-containing species except for 18:0/20:4 1,2-diacylglycerol were significantly decreased. The content of 1,2-diacylglycerol was lowered by 23 and 16% in bovine brain ganglioside and AGF1-treated diabetic animals, respectively, and the quantity of 18:0/20:4 1,2-diacylglycerol was also selectively reduced. Ganglioside administration did not affect the diminished levels of arachidonoyl-containing molecular species in 1,2-diacylglycerol, phosphatidic acid or diacylglycerolipids in nerve from diabetic rats. In the same nerves, bovine brain gangliosides partially and AGF1 completely restored Na+,K(+)-ATPase activity. The results suggest that gangliosides depress the content of total 1,2-diacylglycerol and the quantity of 18:0/20:4 1,2-diacylglycerol, specifically, in diabetic nerve. The possible relationship between the corrective action of gangliosides on Na+,K(+)-ATPase activity and the effect of these substances on 1,2-diacylglycerol molecular species composition and metabolism is discussed.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Diabetes Mellitus, Experimental / enzymology
  • Diabetes Mellitus, Experimental / metabolism*
  • Diglycerides / metabolism*
  • Gangliosides / administration & dosage
  • Gangliosides / pharmacology*
  • Male
  • Ouabain / pharmacology
  • Phosphatidic Acids / metabolism
  • Rats
  • Rats, Sprague-Dawley
  • Sciatic Nerve / drug effects*
  • Sciatic Nerve / enzymology
  • Sciatic Nerve / metabolism
  • Sodium-Potassium-Exchanging ATPase / metabolism

Substances

  • 1,2-diacylglycerol
  • Diglycerides
  • Gangliosides
  • Phosphatidic Acids
  • Ouabain
  • Sodium-Potassium-Exchanging ATPase