Inhalation kinetics of C8 to C10 1-alkenes and iso-alkanes in the rat after repeated exposures

Pharmacol Toxicol. 1993 Sep;73(3):163-8. doi: 10.1111/j.1600-0773.1993.tb01557.x.

Abstract

The toxicokinetic properties of C8 and C10 1-alkenes and iso-alkanes have been investigated in rats during inhalation of 100 p.p.m. of the single hydrocarbons for 3 days, 12 hr/day. The concentration of hydrocarbon was measured in blood, brain, liver, kidneys and perirenal fat at days 1, 2 and 3, immediately after exposure and 12 hr after exposure on day 3. The 1-alkenes showed an efficient absorption to blood combined with extensive accumulation in organs, compared to the iso-alkanes. The concentration of 1-alkenes and iso-alkanes in blood, brain, liver and fat increased with increasing number of carbon atoms. The C9 and C10 1-alkenes and iso-alkanes showed increasing concentration in fat during the exposure period and high concentrations 12 hr after cessation of exposure. The extensive accumulation in both blood and organs of 1-alkenes compared to any of the other groups of hydrocarbons may have a toxicologic relevance. Products which contain 1-alkenes should be handled carefully to minimize the risk of inhalation exposure.

MeSH terms

  • Absorption
  • Adipose Tissue / metabolism
  • Administration, Inhalation
  • Alkanes / administration & dosage
  • Alkanes / chemistry
  • Alkanes / pharmacokinetics*
  • Alkenes / administration & dosage
  • Alkenes / chemistry
  • Alkenes / pharmacokinetics*
  • Animals
  • Brain / metabolism
  • Chromatography, Gas
  • Kidney / metabolism
  • Liver / metabolism
  • Male
  • Rats
  • Rats, Sprague-Dawley
  • Structure-Activity Relationship

Substances

  • Alkanes
  • Alkenes