Suramin selectively inhibits the non-adrenergic non-cholinergic inhibitory junction potential in the guinea-pig stomach

Eur J Pharmacol. 1993 Nov 2;249(1):121-3. doi: 10.1016/0014-2999(93)90671-4.

Abstract

In smooth muscle cells of the guinea-pig stomach fundus, transmural nerve stimulation evoked a cholinergic excitatory junction potential (e.j.p.) and, in the presence of atropine, a non-adrenergic non-cholinergic (NANC) inhibitory junction potential (i.j.p.). Suramin (> 10(-5) M), a putative inhibitor of the P2 purinoceptor, enhanced the e.j.p. amplitude and inhibited the i.j.p., with no significant effect on the membrane potential. Thus, a possible involvement of ATP in the generation of the NANC i.j.p. has to be considered.

MeSH terms

  • Animals
  • Autonomic Nervous System / drug effects
  • Autonomic Nervous System / physiology*
  • Electric Stimulation
  • Gastric Fundus / drug effects*
  • Gastric Fundus / innervation
  • Gastric Fundus / physiology
  • Guinea Pigs
  • Male
  • Membrane Potentials / drug effects
  • Muscle, Smooth / drug effects*
  • Muscle, Smooth / innervation
  • Muscle, Smooth / physiology
  • Neuromuscular Junction / drug effects*
  • Receptors, Purinergic / drug effects
  • Receptors, Purinergic / metabolism
  • Suramin / pharmacology*

Substances

  • Receptors, Purinergic
  • Suramin