Influence of template primary structure on 3'-azido-3'-deoxythymidine triphosphate incorporation into DNA

Antiviral Res. 1993 Jun;21(2):93-102. doi: 10.1016/0166-3542(93)90046-l.

Abstract

In the present study, templates containing a specific segment of the G gamma-globin gene were constructed and incorporation of 3'-azido-3'-deoxythymidine 5'-triphosphate (AZT-TP) or 2',3'-dideoxythymidine 5'-triphosphate (ddTTP) into these templates was compared to that observed in M13 bacteriophage DNA. Investigations on the intrinsic fidelity of T7 DNA polymerase in reactions with AZT-TP and without deoxythymidine 5'-triphosphate, resulted in DNA synthesis beyond the first T site, suggesting that other normal deoxynucleotides misincorporated at these T sites. Modified T7 DNA polymerase incorporated AZT-TP into T sites of elongating DNA strands. Chain termination at noncomplementary sites was also observed with AZT-TP when a genomic DNA template was used and interestingly, this phenomenon was not detected in the presence of a M13 DNA template. These DNA template-dependent effects were not detected with either ddTTP, 2',3'-dideoxycytidine 5'-triphosphate, or 2',3'-didehydro-2',3'-dideoxythymidine 5'-triphosphate (D4T-TP). A variation in the extent of chain termination at T sites was observed with D4T-TP suggesting that each 2',3'-dideoxynucleoside may exhibit unique chain termination patterns along with the template sequence.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Antiviral Agents / metabolism*
  • Bacteriophage M13
  • Base Sequence
  • DNA / metabolism*
  • DNA, Viral / metabolism
  • DNA-Directed DNA Polymerase / metabolism*
  • Dideoxynucleotides
  • Globins / genetics
  • Molecular Sequence Data
  • Substrate Specificity
  • Thymine Nucleotides / metabolism*
  • Zidovudine / analogs & derivatives*
  • Zidovudine / metabolism

Substances

  • Antiviral Agents
  • DNA, Viral
  • Dideoxynucleotides
  • Thymine Nucleotides
  • Zidovudine
  • zidovudine triphosphate
  • Globins
  • DNA
  • bacteriophage T7 induced DNA polymerase
  • DNA-Directed DNA Polymerase