Absorption of zidovudine in patients with diarrhoea

Eur J Clin Pharmacol. 1993;44(5):501-3. doi: 10.1007/BF00315553.

Abstract

Many patients with AIDS have gastrointestinal complaints, including the major clinical disorder of chronic diarrhoea. The pharmacokinetics of zidovudine was studied in 9 male patients with HIV infection and diarrhoea to establish whether drug absorption was impaired in them. The peak plasma concentration and AUC after a single oral dose of 200 mg, were the same as those reported in 6 healthy male volunteers (3.1 vs 4.0 mumol.l-1 and 7.2 vs 5.2 mumol.h.l-1, respectively). Since the bioavailability of zidovudine is not particularly impaired, oral zidovudine therapy can be maintained in patients with diarrhoea.

Publication types

  • Comparative Study

MeSH terms

  • Acquired Immunodeficiency Syndrome / complications
  • Acquired Immunodeficiency Syndrome / metabolism*
  • Adult
  • Biological Availability
  • Chronic Disease
  • Diarrhea / complications
  • Diarrhea / metabolism*
  • Humans
  • Intestinal Absorption*
  • Male
  • Middle Aged
  • Zidovudine / antagonists & inhibitors
  • Zidovudine / pharmacokinetics*

Substances

  • Zidovudine