NK2 receptors mediate plasma extravasation in guinea-pig lower airways

Br J Pharmacol. 1993 Feb;108(2):383-6. doi: 10.1111/j.1476-5381.1993.tb12813.x.

Abstract

1. Neurokinin (NK) receptor-mediated extravasation has been examined in guinea-pig airways by use of a recently described marker for microvascular protein leakage, 125I-labelled human fibrinogen. 2. Neurokinin A (NKA) caused a dose-dependent increase in plasma [125I]-fibrinogen extravasation in trachea, main bronchi, secondary bronchi and intraparenchymal airways. In contrast, the NK2 selective agonist [beta-Ala8]NKA(4-10) only caused extravasation in the secondary and intraparenchymal airways. 3. The NK2 selective antagonist, SR 48968, caused a dose-dependent inhibition of NKA and [beta-Ala8]NKA(4-10)-induced extravasation of fibrinogen in guinea-pig secondary bronchi and intraparenchymal airways. SR 48968 was without effect on the NKA-induced extravasation in trachea and main bronchi. 4. NKA- or [beta-Ala8]NKA(4-10)-induced plasma extravasation was not modified by pretreatment with histamine H1- or H2-receptor antagonists. 5. It is concluded that NK2 receptors mediate plasma [125I]-fibrinogen extravasation in guinea-pig secondary bronchi and intraparenchymal airways. This effect is direct and does not depend upon histamine released from mast cells.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Benzamides / pharmacology*
  • Blood Proteins / metabolism
  • Bronchi / drug effects*
  • Extravasation of Diagnostic and Therapeutic Materials
  • Guinea Pigs
  • Iodine Radioisotopes
  • Male
  • Neurokinin A / analogs & derivatives*
  • Neurokinin A / antagonists & inhibitors*
  • Neurokinin A / pharmacology
  • Peptide Fragments / pharmacology*
  • Piperidines / pharmacology*
  • Receptors, Neurokinin-2
  • Receptors, Neurotransmitter / drug effects
  • Receptors, Neurotransmitter / physiology*

Substances

  • Benzamides
  • Blood Proteins
  • Iodine Radioisotopes
  • Peptide Fragments
  • Piperidines
  • Receptors, Neurokinin-2
  • Receptors, Neurotransmitter
  • neurokinin A (4-10), beta-Ala(8)-
  • SR 48968
  • Neurokinin A