Behavioural and biochemical effects of acute central metabolic inhibition: effects of acetyl-l-carnitine

Eur J Pharmacol. 1993 Apr 28;235(2-3):275-81. doi: 10.1016/0014-2999(93)90146-9.

Abstract

In the present study we evaluated a new method to assess the behavioural and biochemical effects of a brief period of acute hypoxia in the brain. In this method, cyanide is injected into the lateral ventricles. Spatial navigation performance in a Morris task was found to be impaired 1 and 5 min after an i.c.v. injection of 5.0 micrograms cyanide but not after 2.5 micrograms cyanide. Increased rate of phosphatidic acid formation, reflecting increased phospholipase C activity, were observed after injection of 5.0 micrograms cyanide, indicating that energy-dependent phosphoinositide metabolism was affected. Chronic treatment with acetyl-l-carnitine attenuated the cyanide-induced behavioural deficit, but had no effect on energy-dependent phosphoinositide metabolism. The results suggest that, in this model, acetyl-l-carnitine may act via free fatty acid metabolism, by increasing the reservoir of activated acyl groups which are involved in the reacylation of membrane phospholipids.

MeSH terms

  • Acetylcarnitine / pharmacology*
  • Animals
  • Behavior, Animal / drug effects*
  • Brain / drug effects*
  • Brain / metabolism
  • Brain / pathology
  • Chromatography, Thin Layer
  • Cyanides / pharmacology
  • Diglycerides / metabolism
  • Discrimination Learning / drug effects
  • Male
  • Phosphatidylinositols / metabolism
  • Phosphorylation / drug effects
  • Rats
  • Rats, Inbred Strains
  • Subcellular Fractions

Substances

  • Cyanides
  • Diglycerides
  • Phosphatidylinositols
  • Acetylcarnitine