Allosteric modulation by ATP, calcium and magnesium ions of rat osseous plate alkaline phosphatase

Biochim Biophys Acta. 1993 Sep 3;1202(1):22-8. doi: 10.1016/0167-4838(93)90058-y.

Abstract

Alkaline phosphatase from rat osseous plate is allosterically modulated by ATP, calcium and magnesium at pH 7.5. At pH 9.4, the hydrolysis of ATP and PNPP follows Michaelis-Menten kinetics with K0.5 values of 154 microM and 42 microM, respectively. However, at pH 7.5 both substrates exhibit more complex saturation curves, while only ATP exhibited site-site interactions. Ca(2+)-ATP and Mg(2+)-ATP were effective substrates for the enzyme, while the specific activity of the enzyme for the hydrolysis of ATP at pH 7.5 was 800-900 U/mg and was independent of the ion species. ATP, but not PNPP, was hydrolyzed slowly in the absence of metal ions with a specific activity of 140 U/mg. These data demonstrate that in vitro and at pH 7.5 rat osseous plate alkaline phosphatase is an active calcium or magnesium-activated ATPase.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • 4-Nitrophenylphosphatase / metabolism
  • Adenosine Triphosphate / metabolism
  • Adenosine Triphosphate / pharmacology*
  • Alkaline Phosphatase / isolation & purification
  • Alkaline Phosphatase / metabolism*
  • Animals
  • Bone Matrix / enzymology*
  • Calcium / pharmacology*
  • Enzyme Activation
  • Growth Plate / enzymology*
  • Hydrogen-Ion Concentration
  • Kinetics
  • Magnesium / pharmacology*
  • Male
  • Rats
  • Rats, Wistar

Substances

  • Adenosine Triphosphate
  • Alkaline Phosphatase
  • 4-Nitrophenylphosphatase
  • Magnesium
  • Calcium