Effects of beta 6 amino acid hydrophobicity on stability and solubility of hemoglobin tetramers

FEBS Lett. 1993 Jan 2;315(1):47-50. doi: 10.1016/0014-5793(93)81130-r.

Abstract

The relationship between different amino acids at the beta 6 position of hemoglobin and tetramer stability was addressed by a site-directed mutagenesis approach. Precipitation rates during mechanical agitation of oxyhemoglobins with Gln, Ala, Val, Leu and Trp at the beta 6 position increased 2, 5, 13, 21 and 53 times, respectively, compared with that for Hb A. There was a linear relationship between the log of the precipitation rate constant and amino acid hydrophobicity at the beta 6 position, suggesting that enhanced precipitation of oxy Hb S during mechanical agitation results in part from increased hydrophobicity of beta 6 Val. Deoxyhemoglobin solubility increased in the order of beta 6 Ile, Leu, Val, Trp, Gln, Ala and Glu suggesting that hydrophobic interactions between beta 6 Val and the acceptor site of another hemoglobin molecule during deoxy-Hb S polymerization not only depend on hydrophobicity but also on stereospecificity of the amino acid side chain at the beta 6 position. Furthermore, our results indicate that hydrophobic amino acids at the beta 6 position which promote tetramer instability in the oxy form do not necessarily promote polymerization in the deoxy form.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Hemoglobins / chemistry*
  • Humans
  • In Vitro Techniques
  • Mutagenesis, Site-Directed
  • Oxyhemoglobins / chemistry
  • Protein Conformation
  • Protein Denaturation
  • Recombinant Proteins
  • Solubility
  • Stress, Mechanical
  • Structure-Activity Relationship

Substances

  • Hemoglobins
  • Oxyhemoglobins
  • Recombinant Proteins