Isolation and identificaton of an in vivo reaction product of 6-hydroxydopamine

J Med Chem. 1977 Apr;20(4):581-3. doi: 10.1021/jm00214a026.

Abstract

The product of oxidized 6-OHDA and GSH reacted in vitro has been identified by a variety of chemical and physical methods to be 2,4,5-trihydroxy-6-S-(glutathionyl)phenethylamine. Its chemical properties show it easily undergoes a variety of oxidative condensations and polymerization. Its oxidized form, the p-quinone, can be identified in small quantities in rat brain and mouse brain 1-3 h after 6-OHDA injection. This is believed to be the first report of a chemically identified species resulting from the in vivo interaction of 6-OHDA with CNS tissue.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Animals
  • Chemical Phenomena
  • Chemistry
  • Chromatography, High Pressure Liquid
  • Cyclization
  • Glutathione / metabolism
  • Hydroxydopamines / metabolism*
  • Hypothalamus / metabolism
  • Male
  • Mice
  • Oxidation-Reduction
  • Rats
  • Time Factors

Substances

  • Hydroxydopamines
  • Glutathione