Chronic treatment with MK-801 affects the behavioral response to both D1 and D2 dopamine agonist in the one-trial inhibitory avoidance

Psychopharmacology (Berl). 1995 Oct;121(3):401-5. doi: 10.1007/BF02246081.

Abstract

Post-training administration of the N-methyl-D-aspartate (NMDA) antagonists CPP (0.5 and 1.0 mg/kg) and MK-801 (0.25 and 0.5 mg/kg) impaired, in a dose dependent fashion, the one-trial inhibitory avoidance response in NMRI mice. The D1 dopamine (DA) agonist SKF 38393 (10 and 20 mg/kg) and the D2 agonist quinpirole (0.5 and 1.0 mg/kg) instead facilitate the response in the same behavioral paradigm. Sub-chronic blockade of NMDA receptors with MK-801 (0.25 mg/kg once a day for 14 days) did not change the response to both competitive (CPP) and non-competitive (MK-801) NMDA antagonists. The same chronic treatment with MK-801 induced an increased response to both SKF 38393 and quinpirole. These data suggest that repeated administration of MK-801 induce an upregulation of both D1 and D2 DA receptors without affecting NMDA receptors.

MeSH terms

  • 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine / pharmacology
  • Animals
  • Avoidance Learning / drug effects*
  • Behavior, Animal / drug effects*
  • Dizocilpine Maleate / pharmacology*
  • Dopamine Agonists / pharmacology*
  • Dose-Response Relationship, Drug
  • Ergolines / pharmacology
  • Male
  • Mice
  • Mice, Inbred Strains
  • Quinpirole
  • Receptors, Dopamine D1 / agonists
  • Receptors, Dopamine D2 / agonists

Substances

  • Dopamine Agonists
  • Ergolines
  • Receptors, Dopamine D1
  • Receptors, Dopamine D2
  • Quinpirole
  • 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine
  • Dizocilpine Maleate