An insulin peptide that binds an alternative site in class II major histocompatibility complex

J Exp Med. 1996 Mar 1;183(3):857-66. doi: 10.1084/jem.183.3.857.

Abstract

We report that a peptide from the B chain of insulin, B(10-30), binds with high affinity to multiple class II proteins, including IAb,d,k, IEd,k, and DR1. The ability of B(10-30) to inhibit the binding of other peptide antigens to class II does not correlate with its affinity for class II. B(10-30) only weakly inhibits the binding of antigenic peptides. Conversely, peptides with high affinity for the peptide-binding groove of various class II proteins do not inhibit B(10-30) binding. The rate of association of B(10-30) with class II is unusually rapid, approaching saturation in 1-2 h compared with 1-2 d for classical peptide antigens in the same conditions. The dissociation rate is also relatively rapid. The B(10-30) peptide inhibits the binding of the super-antigen staphylococcal enterotoxin B (SEB) to IAk. It also inhibits SEB-mediated T cell activation. These observations support the conclusion that B(10-30) binds to a site outside the peptide-binding groove. Our findings indicate that short-lived peptide-class II complexes can be formed through interactions involving the SEB-binding site and raise the possibility that alternative complexes may serve as T cell receptor ligands.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Binding Sites
  • Binding, Competitive
  • Cattle
  • Cells, Cultured
  • Enterotoxins / toxicity
  • HLA-DR1 Antigen / metabolism*
  • Histocompatibility Antigens Class II / isolation & purification
  • Histocompatibility Antigens Class II / metabolism*
  • Humans
  • Insulin / chemistry
  • Insulin / immunology*
  • Insulin / metabolism
  • Kinetics
  • Lymphocyte Activation
  • Lymphoma, B-Cell
  • Macromolecular Substances
  • Molecular Sequence Data
  • Peptide Fragments / chemistry
  • Peptide Fragments / immunology*
  • Peptide Fragments / pharmacology
  • Staphylococcus aureus
  • Structure-Activity Relationship
  • T-Lymphocytes / drug effects
  • T-Lymphocytes / immunology*

Substances

  • Enterotoxins
  • HLA-DR1 Antigen
  • Histocompatibility Antigens Class II
  • I-E-antigen
  • Insulin
  • Macromolecular Substances
  • Peptide Fragments
  • enterotoxin B, staphylococcal