Mapping of catalytic residues in the RNA polymerase active center

Science. 1996 Jul 5;273(5271):107-9. doi: 10.1126/science.273.5271.107.

Abstract

When the Mg2+ ion in the catalytic center of Escherichia coli RNA polymerase (RNAP) is replaced with Fe2+, hydroxyl radicals are generated. In the promoter complex, such radicals cleave template DNA near the transcription start site, whereas the beta' subunit is cleaved at a conserved motif NADFDGD (Asn-Ala-Asp-Phe-Asp-Gly-Asp). Substitution of the three aspartate residues with alanine creates a dominant lethal mutation. The mutant RNAP is catalytically inactive but can bind promoters and form an open complex. The mutant fails to support Fe2+-induced cleavage of DNA or protein. Thus, the NAD-FDGD motif is involved in chelation of the active center Mg2+.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Aspartic Acid / metabolism
  • Binding Sites
  • DNA / metabolism
  • DNA-Directed RNA Polymerases / chemistry*
  • DNA-Directed RNA Polymerases / genetics
  • DNA-Directed RNA Polymerases / metabolism*
  • Dithiothreitol / pharmacology
  • Electrophoresis, Polyacrylamide Gel
  • Escherichia coli / enzymology*
  • Ferrous Compounds / metabolism
  • Hydroxyl Radical
  • Magnesium / metabolism
  • Molecular Sequence Data
  • Mutagenesis
  • Promoter Regions, Genetic

Substances

  • Ferrous Compounds
  • Aspartic Acid
  • Hydroxyl Radical
  • DNA
  • DNA-Directed RNA Polymerases
  • Magnesium
  • Dithiothreitol