Difference in the mechanism of interaction of Raf-1 and B-Raf with H-Ras

Biochem Biophys Res Commun. 1996 Jun 25;223(3):729-34. doi: 10.1006/bbrc.1996.0964.

Abstract

Ras is known to possess multiple cellular targets including Raf-1. Here, we measured both direct binding of various H-Ras mutants to two representative mammalian Ras targets, Raf-1 and B-Raf, and the activity of the mutants to stimulate Raf-1 and B-Raf, and analysed the difference in their Ras-interaction mechanisms. B-Raf was shown to share almost the same H-Ras binding-specificity with Raf-1 by examining binding of the H-Ras mutants to Raf-1 and B-Raf in the yeast two-hybrid and in vitro binding assays. Mutants, Y32F, A59E, and V45E bound to Raf-1 in Sf9 cells coexpressing them, but failed to activate Raf-1. On the other hand, Y32F activated B-Raf in a cell-free system which consisted of rat brain cytosol and recombinant MEK. These results suggest that there is a subtle structural difference in requirements for the interaction of Ras with Raf-1 and B-Raf.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Brain / metabolism
  • Calcium-Calmodulin-Dependent Protein Kinases / metabolism
  • Cell Line
  • Cytosol / metabolism
  • Genes, ras
  • Kinetics
  • Molecular Sequence Data
  • Point Mutation
  • Protein Serine-Threonine Kinases / metabolism*
  • Proto-Oncogene Proteins / metabolism*
  • Proto-Oncogene Proteins c-raf
  • Proto-Oncogenes
  • Rats
  • Recombinant Proteins
  • Spodoptera
  • Transfection
  • ras Proteins / metabolism*

Substances

  • Proto-Oncogene Proteins
  • Recombinant Proteins
  • Protein Serine-Threonine Kinases
  • Proto-Oncogene Proteins c-raf
  • Calcium-Calmodulin-Dependent Protein Kinases
  • ras Proteins