Mifepristone: antineoplastic studies

Clin Obstet Gynecol. 1996 Jun;39(2):498-505. doi: 10.1097/00003081-199606000-00023.

Abstract

PIP: Emerging research suggests that mifepristone may have significant clinical applications in the treatment of certain neoplastic disorders. For example, in vitro studies have shown that RU-486 can inhibit or stimulate--depending on the cell line and the hormonal milieu of the culture medium--the growth of breast cancer cells. In hormone-sensitive breast cancer, anti-tumor activity is maximized by treatment with a combination of RU-486 and estrogen antagonists such as tamoxifen or luteinizing hormone releasing hormone analogues. The few studies of RU-486 administration in women with advanced breast cancer that had failed to respond to tamoxifen have demonstrated short-term disease stabilization (e.g., 5-10 months). This research has suggested that progesterone receptors are necessary but not sufficient for anti-tumor responses. Also promising, although untested in a large-scale study, is use of RU-486 in women with progressive recurrent and/or unresectable benign meningiomas. In addition, RU-486 has inhibited hormone-insensitive human prostate cancer cell lines grown in vitro and in nude mice xenografts.

Publication types

  • Review

MeSH terms

  • Animals
  • Antineoplastic Agents, Hormonal / pharmacology
  • Antineoplastic Agents, Hormonal / therapeutic use*
  • Breast Neoplasms / drug therapy*
  • Clinical Trials as Topic
  • Female
  • Hormone Antagonists / pharmacology
  • Hormone Antagonists / therapeutic use*
  • Humans
  • Meningeal Neoplasms / drug therapy*
  • Meningioma / drug therapy*
  • Mifepristone / pharmacology
  • Mifepristone / therapeutic use*

Substances

  • Antineoplastic Agents, Hormonal
  • Hormone Antagonists
  • Mifepristone