Effect of leukotriene D4 on tracheal mucociliary transport velocity in quails

Jpn J Pharmacol. 1996 Feb;70(2):195-7. doi: 10.1254/jjp.70.195.

Abstract

We investigated the effect of leukotriene D4 (LTD4) on tracheal mucociliary transport in quails. Topical application of LTD4 (0.2-2 ng) to tracheal mucosa dose-dependently increased mucociliary transport velocity (MCTV) in 5 or 10 min after application. Forty minutes after application of 2 ng of LTD4, MCTV was decreased to about 84% of that in the control group. Both the transient increase and the subsequent decrease induced by 2 ng of LTD4 were blocked by ONO-1078 (Pranlukast: 4-oxo-8-[4-(4-phenylbutoxy)-benzoylamino]-2-(tetrazol-5-yl)- 4H- 1-benzopyran) (0.03-3 mg/kg, i.m.), a specific leukotriene antagonist. These results suggest that LTD4 possesses a biphasic effect on tracheal mucociliary transport through leukotriene receptors.

MeSH terms

  • Animals
  • Dose-Response Relationship, Drug
  • Leukotriene D4 / pharmacology*
  • Male
  • Mucociliary Clearance / drug effects*
  • Quail
  • Time Factors
  • Trachea / drug effects*

Substances

  • Leukotriene D4