Distinct effects of N omega-nitro-L-arginine on seizures induced by several drugs in mice

Pharmacol Biochem Behav. 1996 Mar;53(3):673-7. doi: 10.1016/0091-3057(95)02068-3.

Abstract

A potent nitric oxide (NO) synthase inhibitor, N omega-nitro-L-arginine (L-NA), suppressed tonic seizure elicited by pentylenetetrazol (PTZ; 100 mg/kg, SC) in a dose-related manner (25 to 100 mg/kg, IP), but had no effect on clonic seizure. The effect was most potent at 1 h after the administration of L-NA. L-NA (100 mg/kg, IP) suppressed clonic seizure as well as tonic seizure in bicuculline-treated (3.0 or 4.5 mg/kg, SC) mice. However, it did not affect seizures elicited by picrotoxin (2.0 to 6.0 mg/kg, SC). On the other hand, N-methyl-DL-aspartate (NMDLA; 300 mg/kg or 350 mg/kg, IP) induced clonic seizure, but tonic seizure was not always noted. All mice with clonic and tonic seizures died, and some mice with clonic seizure died without accompanying tonic seizure. L-NA did not influence NMDLA-induced seizures, but it appeared to enhance NMDLA lethality, though without statistical significance. These findings suggest distinct roles of NO in seizures induced by different drugs in mice.

MeSH terms

  • Animals
  • Arginine / analogs & derivatives
  • Arginine / pharmacology*
  • Bicuculline / pharmacology
  • Dose-Response Relationship, Drug
  • Male
  • Mice
  • Mice, Inbred ICR
  • Pentylenetetrazole / pharmacology
  • Picrotoxin / pharmacology
  • Seizures / chemically induced*
  • Time Factors

Substances

  • Picrotoxin
  • Arginine
  • Pentylenetetrazole
  • Bicuculline