Rapid down-regulation of beta-adrenergic receptors evoked by combined forced swimming test and CGP 37849--a competitive antagonist of NMDA receptors

Pol J Pharmacol. 1995 Nov-Dec;47(6):537-40.

Abstract

The influence of CGP 37849, a competitive antagonist of NMDA, receptors and desipramine (DMI) on the density of beta-adrenergic receptors in rats exposed to the forced swimming test was investigated. CGP 37849 (10 mg/kg) and DMI (15 mg/kg), given twice to rats (24 h apart), or the forced swimming test alone failed to alter the density of beta-adrenergic receptors in the rat cortex, as tested using [3H]dihydroalprenolol ([3H]DHA). However, in rats injected with CGP 37849 (10 mg/kg) or DMI (15 mg/kg) and exposed to the forced swimming test, it was found that the density of beta-adrenergic receptors in the cortex was decreased. It was also observed that CGP 37849 used in a dose which decreased the density of beta-adrenergic receptors reduced the immobility time in a manner similar to DMI. It is concluded that CGP 37849 may evoke similar adaptive receptor changes as anti-depressant drugs which-in turn-suggests antidepressant-like properties of CGP 37849.

MeSH terms

  • 2-Amino-5-phosphonovalerate / analogs & derivatives*
  • 2-Amino-5-phosphonovalerate / pharmacokinetics
  • 2-Amino-5-phosphonovalerate / pharmacology
  • Adrenergic Uptake Inhibitors / pharmacology
  • Adrenergic beta-Antagonists / pharmacokinetics
  • Adrenergic beta-Antagonists / pharmacology*
  • Animals
  • Desipramine / pharmacology
  • Dihydroalprenolol
  • Down-Regulation / drug effects*
  • Excitatory Amino Acid Antagonists / pharmacokinetics
  • Excitatory Amino Acid Antagonists / pharmacology*
  • Male
  • Motor Activity / drug effects
  • Rats
  • Rats, Wistar
  • Receptors, Adrenergic, beta / drug effects*
  • Receptors, N-Methyl-D-Aspartate / antagonists & inhibitors*
  • Stress, Psychological / physiopathology*

Substances

  • Adrenergic Uptake Inhibitors
  • Adrenergic beta-Antagonists
  • Excitatory Amino Acid Antagonists
  • Receptors, Adrenergic, beta
  • Receptors, N-Methyl-D-Aspartate
  • 2-amino-4-methyl-5-phosphono-3-pentenoic acid
  • Dihydroalprenolol
  • 2-Amino-5-phosphonovalerate
  • Desipramine