Insulin stimulates mitogen-activated protein kinase by a Ras-independent pathway in 3T3-L1 adipocytes

J Biol Chem. 1996 Nov 29;271(48):30625-30. doi: 10.1074/jbc.271.48.30625.

Abstract

To characterize tissue-specific differences in insulin signaling, we compared the mechanisms of mitogen-activated protein (MAP) kinase activation by insulin in the mitogenically active 3T3-L1 fibroblasts with the metabolically active 3T3-L1 adipocytes. In both cell lines, insulin significantly increased p21(ras).GTP loading (1.5-2-fold) and MAP kinase activity (5-8-fold). Inhibition of Ras farnesylation with lovastatin blocked activation of p21(ras) and Raf-1 kinase in both 3T3-L1 fibroblasts and 3T3-L1 adipocytes. In 3T3-L1 fibroblasts, this was accompanied by an inhibition of the stimulatory effect of insulin on MAP kinase. In contrast, in 3T3-L1 adipocytes, despite an inhibition of activation of p21(ras) and Raf-1 by lovastatin, insulin continued to stimulate MAP kinase activity. Fractionation of the cell lysates on the FPLC Mono-Q column revealed that lovastatin inhibited insulin stimulation of ERK2 (and, to a lesser extent, ERK1) in 3T3-L1 fibroblasts and had no effect on the insulin-stimulated ERK2 in 3T3-L1 adipocytes. These results demonstrate an important distinction between the mechanism of insulin signaling in the metabolically and mitogenically active cells. Insulin activates MAP kinase by the Ras-dependent pathway in the 3T3-L1 fibroblasts and by the Ras-independent pathway in the 3T3-L1 adipocytes.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Adipocytes / enzymology*
  • Alkyl and Aryl Transferases*
  • Animals
  • Calcium-Calmodulin-Dependent Protein Kinases / metabolism*
  • Enzyme Activation / drug effects
  • Enzyme Inhibitors / pharmacology
  • Farnesol / analogs & derivatives
  • Farnesol / pharmacology
  • Farnesyltranstransferase
  • Guanosine Triphosphate / metabolism
  • Hydroxymethylglutaryl-CoA Reductase Inhibitors
  • Insulin / pharmacology*
  • Lovastatin / pharmacology
  • Mice
  • Organophosphonates*
  • Organophosphorus Compounds / pharmacology
  • Protein Kinase C / physiology
  • Protein Serine-Threonine Kinases / metabolism
  • Proto-Oncogene Proteins / metabolism
  • Proto-Oncogene Proteins c-raf
  • Proto-Oncogene Proteins p21(ras) / physiology
  • Rats
  • Signal Transduction
  • Transferases / antagonists & inhibitors

Substances

  • (alpha-hydroxyfarnesyl)phosphonic acid
  • Enzyme Inhibitors
  • Hydroxymethylglutaryl-CoA Reductase Inhibitors
  • Insulin
  • Organophosphonates
  • Organophosphorus Compounds
  • Proto-Oncogene Proteins
  • Farnesol
  • Guanosine Triphosphate
  • Lovastatin
  • Transferases
  • Alkyl and Aryl Transferases
  • Farnesyltranstransferase
  • Protein Serine-Threonine Kinases
  • Proto-Oncogene Proteins c-raf
  • Protein Kinase C
  • Calcium-Calmodulin-Dependent Protein Kinases
  • Proto-Oncogene Proteins p21(ras)