Angiotensin II, via an action at AT1 receptors, may modulate the behavioural effects of ET-1 in conscious rats

Life Sci. 1996;59(22):PL355-8. doi: 10.1016/s0024-3205(96)00541-3.

Abstract

The injection of endothelin-1 (ET-1) (1 pmol/rat) into the dorsolateral periaqueductal gray (PAG) area of freely moving rats induced rotation along the long axis of the body (barrel-rolling). Preinjection (10 min before) of losartan (a selective AT1 receptor antagonist; 50 nmol) to the PAG area reduced the behavioural response to ET-1. In contrast, pretreatment with PD123319 (a selective AT2 receptor antagonist; 50 nmol) did not affect the ET-1-induced barrel-rolling. These results indicate that endogenous angiotensin II, via an action on AT1 receptors, contributes to the barrel-rolling of ET-1 within the brain.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Angiotensin I / metabolism*
  • Angiotensin II / pharmacology*
  • Angiotensin Receptor Antagonists*
  • Animals
  • Behavior, Animal / drug effects*
  • Biphenyl Compounds / pharmacology
  • Drug Synergism
  • Endothelin-1 / pharmacology*
  • Imidazoles / pharmacology
  • Losartan
  • Male
  • Pyridines / pharmacology
  • Rats
  • Rats, Sprague-Dawley
  • Receptors, Angiotensin / metabolism
  • Tetrazoles / pharmacology

Substances

  • Angiotensin Receptor Antagonists
  • Biphenyl Compounds
  • Endothelin-1
  • Imidazoles
  • Pyridines
  • Receptors, Angiotensin
  • Tetrazoles
  • Angiotensin II
  • PD 123319
  • Angiotensin I
  • Losartan