Valence selectivity of the gramicidin channel: a molecular dynamics free energy perturbation study

Biophys J. 1996 Dec;71(6):3177-85. doi: 10.1016/S0006-3495(96)79511-5.

Abstract

The valence selectivity of the gramicidin channel is examined using computer simulations based on atomic models. The channel interior is modeled using a gramicidin-like periodic poly (L,D)-alanine beta-helix. Free energy perturbation calculations are performed to obtain the relative affinity of K+ and Cl- for the channel. It is observed that the interior of the gramicidin channel provides an energetically favorable interaction site for a cation but not for an anion. Relative to solvation in bulk water, the carbonyl CO oxygens can provide a favorable interaction to stabilize K+, whereas the amide NH hydrogens are much less effective in stabilizing Cl-. The results of the calculations demonstrate that, as a consequence of the structural asymmetry of the backbone charge distribution, a K+ cation can partition spontaneously from bulk water to the interior of the gramicidin channel, whereas a Cl- anion cannot.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Calorimetry
  • Chlorides
  • Computer Simulation
  • Gramicidin*
  • Ion Channels*
  • Models, Biological
  • Peptides / chemistry*
  • Potassium
  • Protein Structure, Secondary*
  • Software
  • Thermodynamics

Substances

  • Chlorides
  • Ion Channels
  • Peptides
  • Gramicidin
  • polyalanine
  • Potassium