[The clinicopharmacological case (5). serotonin reuptake inhibitor and 5-HT3-receptor antagonists: are there clinically relevant interactions?]

Praxis (Bern 1994). 1996 Nov 12;85(46):1490-2.
[Article in German]

Abstract

We describe a patient with chronic depression who was treated with the selective serotonin-reuptake-inhibitor sertraline. Following surgery, the patient developed severe nausea and vomiting, necessitating an efficient antiemetic treatment, possibly including the 5-HT3-receptor antagonist ondansetrone. Because both drugs, sertraline and ondansetrone, interact with the serotonin system at the synapsis, a possible interaction was discussed. Since the effect of the selective serotonin-reuptake inhibitors mainly depends on 5-HT1 and 5-HT2-receptors, a pharmacodynamic interaction between an 5-HT3-antagonist and a serotonin-reuptake-inhibitor at the synapsis leading to the relapse of depression seems to be very unlikely. There exist also no conclusive data suggesting a clinically relevant pharmacokinetic interaction between the two drugs. A treatment with ondansetrone was considered to be safe in this patient.

Publication types

  • Case Reports
  • English Abstract

MeSH terms

  • 1-Naphthylamine / analogs & derivatives*
  • 1-Naphthylamine / pharmacology
  • 1-Naphthylamine / therapeutic use
  • Antidepressive Agents / pharmacology
  • Antidepressive Agents / therapeutic use
  • Antiemetics / pharmacology
  • Antiemetics / therapeutic use
  • Depression / drug therapy*
  • Drug Interactions
  • Female
  • Humans
  • Ondansetron / pharmacology
  • Ondansetron / therapeutic use*
  • Receptors, Serotonin / drug effects
  • Selective Serotonin Reuptake Inhibitors / pharmacology
  • Selective Serotonin Reuptake Inhibitors / therapeutic use*
  • Serotonin Antagonists / pharmacology
  • Serotonin Antagonists / therapeutic use*
  • Sertraline

Substances

  • Antidepressive Agents
  • Antiemetics
  • Receptors, Serotonin
  • Serotonin Antagonists
  • Serotonin Uptake Inhibitors
  • Ondansetron
  • 1-Naphthylamine
  • Sertraline