Ras-dependent, Ca2+-stimulated activation of nuclear factor of activated T cells by a constitutively active Cbl mutant in T cells

J Biol Chem. 1997 Jan 3;272(1):168-73. doi: 10.1074/jbc.272.1.168.

Abstract

T cell receptor (TCR) stimulation induces rapid tyrosine phosphorylation of cellular proteins, including Cbl, a protooncogene product whose function remains unclear. As a first step toward elucidating the function of Cbl in TCR-initiated signaling, we evaluated the ability of wild-type Cbl or a transforming Cbl mutant (70Z/3) to induce transcriptional activation of a nuclear factor of activated T cells (NFAT) element derived from the interleukin 2 (IL2) promoter in transiently cotransfected Jurkat-TAg T cells. 70Z/3, but not Cbl, caused NFAT activation which was significantly enhanced by stimulation with calcium ionophore, and was drastically reduced by cyclosporin A pretreatment. A point mutation of a potential phosphatidylinositol 3-kinase (PI3-K) binding site (Y731EAM to Y731EAC) in 70Z/3 disrupted the association of PI3-K with 70Z/3, but did not reduce the induction of NFAT activity, suggesting that the interaction between Cbl and PI3-K is not required in the 70Z/3-mediated induction of NFAT. Additional mapping studies indicated that defined deletions of C-terminal 70Z/3 sequences affected to a variable degree its ability to stimulate NFAT activity. Strikingly, deletion of 346 C-terminal residues augmented this activity, whereas removal of 20 additional residues abolished it. Coexpression of dominant negative Ras abrogated the basal or ionomycin-stimulated, 70Z/3-mediated NFAT activation, suggesting a functional Ras is required for this activation. These results implicate Cbl in Ras-dependent signaling pathways which lead to NFAT activation.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Animals
  • Calcineurin
  • Calcium / physiology*
  • Calmodulin-Binding Proteins / physiology
  • DNA-Binding Proteins / physiology*
  • Humans
  • Ionomycin / pharmacology
  • Lymphocyte Activation
  • Mice
  • NFATC Transcription Factors
  • Nuclear Proteins*
  • Oncogene Protein v-cbl
  • Phosphatidylinositol 3-Kinases
  • Phosphoprotein Phosphatases / physiology
  • Phosphotransferases (Alcohol Group Acceptor) / physiology
  • Proto-Oncogene Proteins / chemistry
  • Proto-Oncogene Proteins / physiology*
  • Proto-Oncogene Proteins c-cbl
  • Proto-Oncogene Proteins p21(ras) / physiology*
  • Retroviridae Proteins, Oncogenic / metabolism
  • Sequence Deletion
  • Structure-Activity Relationship
  • T-Lymphocytes / metabolism*
  • Transcription Factors / physiology*
  • Tumor Cells, Cultured
  • Ubiquitin-Protein Ligases*

Substances

  • Calmodulin-Binding Proteins
  • DNA-Binding Proteins
  • NFATC Transcription Factors
  • Nuclear Proteins
  • Oncogene Protein v-cbl
  • Proto-Oncogene Proteins
  • Retroviridae Proteins, Oncogenic
  • Transcription Factors
  • Ionomycin
  • Proto-Oncogene Proteins c-cbl
  • Ubiquitin-Protein Ligases
  • Phosphatidylinositol 3-Kinases
  • Phosphotransferases (Alcohol Group Acceptor)
  • Calcineurin
  • Phosphoprotein Phosphatases
  • HRAS protein, human
  • Proto-Oncogene Proteins p21(ras)
  • CBL protein, human
  • Cbl protein, mouse
  • Calcium