CFTR-like chloride channels in non-ciliated bronchiolar epithelial (Clara) cells

Biochem Biophys Res Commun. 1997 Jan 13;230(2):470-5. doi: 10.1006/bbrc.1996.5939.

Abstract

Distal airways are believed to be a major site of disease in cystic fibrosis. The product of the CF gene, CFTR, is expressed in non-ciliated bronchiolar epithelial (Clara) cells. Clara cells in primary culture are capable of Cl- secretion which can be stimulated by cAMP and extracellular nucleotides. We used the patch clamp technique to look for Cl- channels in the apical membrane of rabbit Clara cells. In cell-attached patches, we recorded Cl- channels with a conductance for outward currents of 7.5 +/- 0.4 pS (n = 10) and for inward currents of 3.2 +/- 0.5 pS (n = 10); these channels typically exhibited slow kinetics and were not inhibited by the Cl- channel blockers NPPB and DIDS. Channel activity was not noticeably dependent on pipette potential. Addition of chlorophenylthio-cyclic AMP (cpt-cAMP) to the bath increased the percentage of cell-attached patches with active channels (33.8% vs 56.7%; p< 0.05) and the channel open probability (0.49 +/- 0.03 vs 0.84 +/- 0.02; p< 0.05). Extracellular ATP increased the percentage of cell-attached patches with active channels (28.7% to 50.0%; p< 0.05) but had no significant effect on the channel open probability (0.62 +/- 0.07 vs 0.60 +/- 0.06). In conclusion, rabbit non-ciliated bronchiolar epithelial cells express low-conductance Cl- channels that share many similarities with the CFTR-related Cl- channel and are regulated by cAMP and extracellular ATP.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid / pharmacology
  • Adenosine Triphosphate / pharmacology
  • Animals
  • Bronchi / physiology*
  • Cell Membrane / physiology
  • Cells, Cultured
  • Chloride Channels / physiology*
  • Cyclic AMP / analogs & derivatives
  • Cyclic AMP / pharmacology
  • Cystic Fibrosis Transmembrane Conductance Regulator / drug effects
  • Cystic Fibrosis Transmembrane Conductance Regulator / physiology*
  • Electric Conductivity
  • Epithelium / physiology
  • Membrane Potentials / drug effects
  • Nitrobenzoates / pharmacology
  • Patch-Clamp Techniques
  • Rabbits
  • Thionucleotides / pharmacology

Substances

  • Chloride Channels
  • Nitrobenzoates
  • Thionucleotides
  • Cystic Fibrosis Transmembrane Conductance Regulator
  • 5-nitro-2-(3-phenylpropylamino)benzoic acid
  • 8-((4-chlorophenyl)thio)cyclic-3',5'-AMP
  • Adenosine Triphosphate
  • Cyclic AMP
  • 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid