A reductive acidolysis final deprotection strategy in solid phase peptide synthesis based on safety-catch protection

Chem Pharm Bull (Tokyo). 1997 Jan;45(1):18-26. doi: 10.1248/cpb.45.18.

Abstract

A reductive acidolysis final deprotection strategy in solid phase peptide synthesis was developed using a new safety-catch type of semi-permanent protecting groups and new linkers which were derived from 4-methylsulfinylbenzyl protection. This new strategy was based on a two-dimensional protection scheme employing acid-labile temporary and acid-stable but reductive acidolysis-cleavable semi-permanent protecting groups. By using this strategy, we successfully synthesized four model peptides, of which two contained C-terminal amide.

MeSH terms

  • Amino Acid Sequence
  • Molecular Sequence Data
  • Peptides / chemical synthesis*
  • Peptides / chemistry

Substances

  • Peptides