Pentoxifylline, a drug with rheological effects, decreases portal pressure in an experimental model of cirrhosis

Eur J Gastroenterol Hepatol. 1997 Jan;9(1):27-31. doi: 10.1097/00042737-199701000-00009.

Abstract

Objective: To evaluate the influences of blood viscosity changes, mediated by a haemorheological agent, on splanchnic and systemic haemodynamic parameters in rats with cirrhosis due to chronic bile duct ligation.

Methods: Blood viscosity was measured using a cone-plate viscometer and whole blood filterability was determined by a filtration method. Cardiac index and portal venous inflow were measured using radioactive microspheres. Measurements were performed 30 min after double-blind administration of placebo or pentoxifylline (25 mg/kg, intravenously).

Results: As compared with placebo, pentoxifylline-treated cirrhotic rats had a lower portal pressure (13.8 +/- 1.4 vs. 12.1 +/- 1.6 mmHg, P < 0.05) and blood viscosity at shear rates of 115/s (6.6 +/- 0.8 vs. 5.8 +/- 0.3 mPas, P < 0.05), associated with an improvement of whole blood filterability (45.0 +/- 12.9 vs. 20.0 = 3.9 s/ml, P < 0.01). Similar values of mean arterial pressure, cardiac index and portal venous inflow were observed in both groups. A significant correlation was found between portal pressure and blood viscosity at a shear rate of 115/s (r = 0.71, P < 0.01).

Conclusion: These results suggest that portal pressure can be modified by pentoxifylline in an experimental model of cirrhosis. These haemodynamic changes are associated with a lower blood viscosity and whole blood filterability. Pentoxifylline may be a new approach in the treatment of portal hypertension.

Publication types

  • Comparative Study

MeSH terms

  • Animals
  • Blood Viscosity / drug effects
  • Cardiac Output / drug effects
  • Cholestasis / complications
  • Disease Models, Animal
  • Double-Blind Method
  • Hypertension, Portal / drug therapy*
  • Hypertension, Portal / etiology
  • Hypertension, Portal / physiopathology
  • Infusions, Intravenous
  • Liver Cirrhosis, Experimental / complications*
  • Liver Cirrhosis, Experimental / physiopathology
  • Male
  • Pentoxifylline / administration & dosage
  • Pentoxifylline / pharmacology*
  • Portal Pressure / drug effects
  • Rats
  • Rats, Wistar
  • Vasodilator Agents / administration & dosage
  • Vasodilator Agents / pharmacology*

Substances

  • Vasodilator Agents
  • Pentoxifylline