Antitumor effect of CPT-11, a camptothecin derivative, on human testicular tumor xenografts in nude mice

Eur Urol. 1997;31(1):92-6. doi: 10.1159/000474425.

Abstract

Objective: The antitumor effect of CPT-11, a camptothecin derivative, on two human testicular embryonal carcinomas (TTSC-2 and TTSC-3) heterotransplanted into-nude mice was studied.

Materials and methods: Tumor-bearing nude mice were given daily intraperitoneal injections of the anticancer drugs in 0.1 ml saline 3 times at 3-day intervals. At the end of the experiments tumors were resected and subjected to light-microscopic observation.

Results: When 10, 30 and 50 mg/kg of CPT-11 was administered to tumor-bearing mice intraperitoneally, the antitumor effect of CPT-11 was observed dose-dependently in both TTSC-2 and TTSC-3. When 30 mg/kg of CPT-11 was administered in combination with CDDP, complete tumor regression was observed in both TTSC-2 and TTSC-3 tumors. Histological findings correlated well with the decrease in tumor volume of treated tumors. No mice died after treatment with CPT-11 in a single-agent and combination chemotherapy.

Conclusion: Chemotherapy with CPT-11 was an effective and safe method against human testicular tumors heterotransplanted in nude mice.

MeSH terms

  • Animals
  • Antineoplastic Agents / administration & dosage
  • Antineoplastic Agents, Phytogenic / administration & dosage
  • Antineoplastic Agents, Phytogenic / therapeutic use*
  • Antineoplastic Combined Chemotherapy Protocols / therapeutic use
  • Camptothecin / administration & dosage
  • Camptothecin / analogs & derivatives*
  • Camptothecin / therapeutic use
  • Carboplatin / administration & dosage
  • Carboplatin / analogs & derivatives
  • Cisplatin / administration & dosage
  • Dose-Response Relationship, Drug
  • Etoposide / administration & dosage
  • Humans
  • Irinotecan
  • Male
  • Mice
  • Mice, Inbred BALB C
  • Mice, Nude
  • Neoplasm Transplantation
  • Organoplatinum Compounds / administration & dosage
  • Teratocarcinoma / drug therapy*
  • Testicular Neoplasms / drug therapy*
  • Topoisomerase I Inhibitors
  • Transplantation, Heterologous
  • Vinblastine / administration & dosage

Substances

  • Antineoplastic Agents
  • Antineoplastic Agents, Phytogenic
  • Organoplatinum Compounds
  • Topoisomerase I Inhibitors
  • DWA 2114
  • Vinblastine
  • Etoposide
  • Irinotecan
  • nedaplatin
  • Carboplatin
  • Cisplatin
  • Camptothecin