The anxiolytic-like effect of metabotropic glutamate receptor antagonists after intrahippocampal injection in rats

Eur J Pharmacol. 1997 Jan 29;319(2-3):153-6. doi: 10.1016/s0014-2999(96)00941-7.

Abstract

Using the conflict drinking Vogel test in rats as a model we examined the anxiolytic-like activity, after their intrahippocampal administration of (S)-4-carboxy-3-hydroxyphenyl-glycine (S-4C3H-PG), RS-alpha-methylserine-O-phosphate-monophenyl ester (MSOPPE) and (RS)-alpha-methylserine-O-phosphate (MSOP), the antagonists of the I, the II and the III group of metabotropic glutamate receptors (mGlu receptors), respectively. The results indicate that S-4C3H-PG and MSOP produced a dose-dependent anticonflict effect in rats, which was unrelated to a reduced perception of the stimulus or to an increased thirst drive. The hippocampus may be one of the neuroanatomical sites of the anxiolytic-like effects of both mGlu receptor antagonists.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anti-Anxiety Agents / administration & dosage
  • Anti-Anxiety Agents / pharmacology*
  • Conflict, Psychological
  • Drinking / drug effects
  • Drinking Behavior / drug effects
  • Electroshock
  • Excitatory Amino Acid Antagonists / administration & dosage
  • Excitatory Amino Acid Antagonists / pharmacology*
  • Hippocampus / anatomy & histology
  • Hippocampus / drug effects
  • Hippocampus / physiology*
  • Injections
  • Male
  • Rats
  • Rats, Wistar
  • Receptors, Metabotropic Glutamate / antagonists & inhibitors*

Substances

  • Anti-Anxiety Agents
  • Excitatory Amino Acid Antagonists
  • Receptors, Metabotropic Glutamate