Hydrogen exchange in the lipid bilayer-bound gramicidin channel

Solid State Nucl Magn Reson. 1996 Dec;7(3):177-83. doi: 10.1016/s0926-2040(96)01260-x.

Abstract

Hydrogen exchange experiments for a membrane-bound polypeptide could lead to interesting functional and structural insights. Here, hydrogen/deuterium exchange, saturation transfer and differential relaxation experiments have been performed on oriented lipid bilayer-bound polypeptide samples to measure the exchange lifetimes. The polypeptide, gramicidin A, forms a monovalent cation selective channel across membranes. The pH dependent results suggest that the indole N epsilon 1-H groups show base catalyzed hydrogen exchange, but that the backbone amide sites are not base catalyzed, consistent with the exclusion of anions from this channel. Furthermore, the recently described [1] orientational distribution of the individual peptide carbonyls (i.e. carbonyls either tipped slightly in toward or away from the channel axis) is consistent with the observed difference in odd- and even-numbered amide residue exchange lifetimes.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Deuterium
  • Gramicidin / chemistry*
  • Gramicidin / metabolism
  • Hydrogen
  • Hydrogen-Ion Concentration
  • Ion Channels / chemistry*
  • Ion Channels / metabolism
  • Kinetics
  • Lipid Bilayers / chemistry*
  • Lipid Bilayers / metabolism
  • Magnetic Resonance Spectroscopy / methods

Substances

  • Ion Channels
  • Lipid Bilayers
  • Gramicidin
  • Hydrogen
  • Deuterium