Bactericidal activity of DU-6859a compared to activities of three quinolones, three beta-lactams, clindamycin, and metronidazole against anaerobes as determined by time-kill methodology

Antimicrob Agents Chemother. 1997 Apr;41(4):847-9. doi: 10.1128/AAC.41.4.847.

Abstract

The activities of DU-6859a, ciprofloxacin, levofloxacin, sparfloxacin, piperacillin, piperacillin-tazobactam, imipenem, clindamycin, and metronidazole against 11 anaerobes were tested by the broth microdilution and time-kill methods. DU-6859a was the most active drug tested (broth microdilution MICs, 0.06 to 0.5 microg/ml), followed by imipenem (MICs, 0.002 to 4.0 microg/ml). Broth macrodilution MICs were within 3 (but usually 1) dilutions of the broth microdilution MICs. All compounds were bactericidal at the MIC after 48 h; after 24 h, 90% killing was shown for all strains when the compounds were used at four times the MIC. DU-6859a at < or = 0.5 microg/ml was bactericidal after 48 h.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Anti-Bacterial Agents / pharmacology
  • Bacteria, Anaerobic / drug effects*
  • Clindamycin / pharmacology
  • Culture Media
  • Fluoroquinolones*
  • Metronidazole / pharmacology
  • Microbial Sensitivity Tests
  • Quinolones / pharmacology*
  • Time Factors
  • beta-Lactams

Substances

  • Anti-Bacterial Agents
  • Culture Media
  • Fluoroquinolones
  • Quinolones
  • beta-Lactams
  • Metronidazole
  • Clindamycin
  • sitafloxacin