Oligomerization of the soluble granulocyte-macrophage colony-stimulating factor receptor: identification of the functional ligand-binding species

Cytokine. 1997 Apr;9(4):219-25. doi: 10.1006/cyto.1996.0157.

Abstract

The ligand-specific alpha subunit of the dimeric human GM-CSF receptor exists in both transmembrane anchored (tmGM-CSFR alpha) and soluble (sGM-CSFR alpha) isoforms. sGM-CSFR alpha binds to GM-CSF in solution and antagonizes GM-CSF biological activity in vitro. In an effort to better understand the biological properties of sGM-CSFR alpha the authors have attempted to define the exact stoichiometry of the interaction between GM-CSF and sGM-CSFR alpha. Size separation of sGM-CSFR alpha by polyacrylamide gel electrophoresis (PAGE) under non-reducing conditions demonstrated that sGM-CSFR alpha can exist in solution not only in a monomeric state but also in higher order oligomers. FPLC analysis of ligand/sGM-CSFR alpha complexes suggested that only one of these sGM-CSFR alpha species could functionally bind GM-CSF. PAGE analysis of FPLC fractions demonstrated that the peak of GM-CSF binding activity corresponded to the presence of a monomeric form of sGM-CSFR alpha. The experiments demonstrate that while sGM-CSFR alpha can adopt oligomeric forms in solution, the binding of GM-CSF to sGM-CSFR alpha most likely occurs in a (GM-CSF)1 (sGM-CSFR alpha)1 configuration.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Autoradiography
  • Blotting, Western
  • Cell Line
  • Chromatography, High Pressure Liquid
  • Cricetinae
  • Densitometry
  • Electrophoresis, Polyacrylamide Gel
  • Granulocyte-Macrophage Colony-Stimulating Factor / chemistry*
  • Granulocyte-Macrophage Colony-Stimulating Factor / metabolism*
  • Humans
  • Ligands
  • Molecular Structure
  • Protein Binding
  • Receptors, Granulocyte-Macrophage Colony-Stimulating Factor / chemistry*
  • Receptors, Granulocyte-Macrophage Colony-Stimulating Factor / metabolism*
  • Receptors, Granulocyte-Macrophage Colony-Stimulating Factor / physiology
  • Solubility
  • Solutions
  • Structure-Activity Relationship

Substances

  • Ligands
  • Receptors, Granulocyte-Macrophage Colony-Stimulating Factor
  • Solutions
  • Granulocyte-Macrophage Colony-Stimulating Factor