Analysis of the ability of 12-O-tetradecanoylphorbol-13-acetate to induce epidermal hyperplasia, transforming growth factor-alpha, and skin tumor promotion in wa-1 mice

J Invest Dermatol. 1997 May;108(5):784-91. doi: 10.1111/1523-1747.ep12292237.

Abstract

Wa-1 mutant mice possess a defect in the production of transforming growth factor-alpha (TGF-alpha) that leads to a phenotype characterized by wavy hair and curly whiskers. In light of recent evidence indicating the importance of TGF-alpha in epithelial tumorigenesis, this study characterizes the responsiveness of wa-1 mice to skin tumor promotion by the phorbol ester, 12-O-tetradecanoylphorbol-13-acetate (TPA). The responsiveness of wa-1 mice to TPA was compared with that of SENCAR and C57BL/6 mice, representing mouse lines highly sensitive and resistant to skin tumor promotion, respectively. Wa-1 mice were found to be very resistant to skin tumor promotion by TPA after initiation with 10 nmol DMBA, similar to C57BL/6 mice. TPA failed to induce a dramatic increase in TGF-alpha mRNA and protein in the skin of wa-1 mice, whereas TGF-alpha mRNA and protein were dramatically induced in the skin (both epidermis and dermis) of SENCAR and C57BL/6 mice. TPA treatment dramatically increased mRNA levels of two other EGF receptor ligands, amphiregulin and heparin binding-EGF, however, in the skin of all three mouse lines. Comparison of histologic changes in skin revealed that wa-1 mice exhibited only modest sustained epidermal hyperplasia after multiple treatments with TPA, similar in magnitude to that of C57BL/6 mice and significantly lower than that of SENCAR mice. The current data indicate that wa-1 mice are relatively resistant to TPA promotion. Possible mechanisms for this resistance are discussed.

Publication types

  • Comparative Study
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amphiregulin
  • Animals
  • Antineoplastic Agents / metabolism
  • Carcinogens / pharmacology*
  • EGF Family of Proteins
  • Epidermal Growth Factor / metabolism
  • Female
  • Glycoproteins / metabolism
  • Growth Substances / metabolism
  • Heparin / metabolism
  • Heparin-binding EGF-like Growth Factor
  • Hyperplasia / chemically induced
  • Intercellular Signaling Peptides and Proteins*
  • Male
  • Mice
  • Mice, Inbred C57BL / physiology
  • Mice, Inbred SENCAR
  • Mice, Mutant Strains / physiology*
  • Neutrophils / drug effects
  • Neutrophils / physiology
  • RNA, Messenger / metabolism
  • Skin / pathology*
  • Skin Neoplasms / chemically induced*
  • Tetradecanoylphorbol Acetate / pharmacology*
  • Transforming Growth Factor alpha / biosynthesis*
  • Transforming Growth Factor alpha / genetics

Substances

  • Amphiregulin
  • Antineoplastic Agents
  • Areg protein, mouse
  • Carcinogens
  • EGF Family of Proteins
  • Glycoproteins
  • Growth Substances
  • Hbegf protein, mouse
  • Heparin-binding EGF-like Growth Factor
  • Intercellular Signaling Peptides and Proteins
  • RNA, Messenger
  • Transforming Growth Factor alpha
  • Epidermal Growth Factor
  • Heparin
  • Tetradecanoylphorbol Acetate